Product Name:   2- [6-(4-Chloro-phenyl)-1-Methyl-4H-3-oxa-2,5-diaza-benzo[e]azulen-4-yl]-acetaMide

Synonyms: 2-[6-(4-Chloro-phenyl)-1-Methyl-4H-3-oxa-2,5-diaza-benzo[e]azulen-4-yl]-acetaMide; BET bromodomain inhibitor; 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide; CPI-0610; (4S)-6-(4-Chlorophenyl)-1-methyl-4H-isoxazolo[5,4-d][2]benzazepine-4-acetamide; CPI0160

CAS No.: 1380087-89-7

Purity:  98%

Formula: C20H16ClN3O2

Molecular Weight: 365.8

Appearance:  white or off-white Power

Density:  1.41±0.1 g/cm3

Boiling point:  622.8±55.0 °C

Grade: Pharmaceutical Grade

Applications: used as an important raw material and Pharmaceutical intermediates

Package: 1kg/25kg or as client’s requirement

Storage:  avoid light, ventilation and shade

          Power         -20°C     3 years

                    4°C      2 years

Pelabresib (CPI-0610) is a potent, selective, orally active and cell-active BET inhibitor. Pelabresib inhibits BRD4-BD1 with an IC50 of 39 nM, and with an EC50 value of 0.18 μM for MYC.

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